Adrián García Recio - 6.1.
Alejandro Peralta-García - 4.5.
Aleix Quintana - 4.3.
Anna Chorianopoulou - 6.4.
Anna Grimm - 4.7.
Antonio Capó Quetglas - 6.8.
Berta Carrasco Martinez - 5.1.
Bert Beerkens - 1.5.
Camilla Guccione - 2.7.
Charlotte Crauwels - 6.2.
Clizia Russotto - 4.1.
Cristian Lombo - 5.8.
David Aranda - 6.6.
David Shi - 6.5.
Estefanía Moreno - 5.7.
Florian Bößl - 2.5.
Francesco Ferri - 2.2.
Francesco Fontanive - 4.2.
Friederike Wunsch - 1.6.
Hongyue Liu - 6.3.
Jaume Lillo - 2.6.
Joan Biel Rebassa Palou - 5.6.
Judith Alenfelder - 5.3.
Julie Delaroche - 3.7.
Kristoffer Sahlholm - 3.2.
Lucía González-Pico - 5.4.
Marija Popović-Nikolić - 3.8.
Maria Majellaro - 1.3.
Maris-Johanna Tahk - 3.3.
Marc Ciruela Jardí - 2.3.
Marta López Balastegui - 4.4.
Matteo Pavan - 3.5.
Noemi Karsai - 1.4.
Noureldine Youssef - 1.2.
Owen Underwood - 5.5.
Paola Oliva - 4.6.
Paulina Dragan - 1.7.
Petra Ferjan - 2.1.
Ramilya Murtazina - 3.4.
Sadaf Dadashkhan - 1.8.
Shanshan Li - 6.7.
Shubham Vishnoi - 5.2.
Thomas Tarenzi - 3.1.
Tomasz Stepniewski - 3.6.
Wijnand van der Velden - 2.4.
Yao Yao - 1.1.
Poster presentations on November 25, 2024 will be live streamed from 15:50 to 16:20 CET.
Poster 1.5.
Bert Beerkens
Development of an irreversible allosteric probe for investigations towards the CC chemokine receptor 2
Poster 1.2.
Noureldine Youssef
Characterization of distinct GRK requirements and β-arrestin2 conformational changes induced by natural and synthetic ACKR3 agonists
Poster 1.3.
Maria Majellaro
Integrating Binding and Functional Assays for Comprehensive GPCR Screening: CXCR4 Receptor case study
Poster 1.7.
Paulina Dragan
AI-driven GPCRVS in Drug Design Targeting CC, CXC, and Atypical Chemokine Receptors
Poster 1.4.
Noemi Karsai
Ligand-induced changes in the plasma membrane organisation of the chemokine receptor ACKR3
Poster 1.8.
Sadaf Dadashkhan
Calcium ions modulate the activation of metabotropic glutamate receptor by glutamate
Poster presentations on November 25, 2024 will be live streamed from 18:50 to 19:20 CET.
Poster 2.1.
Petra Ferijan
Expression of ADGRA3 in Porcine Ovaries: Insights from Immunohistochemistry and qPCR Analysis
Poster 2.3.
Marc Ciruela Jardí
Design of small, nonpeptidic, ligands to disrupt CB1R-5HT2AR heteromerization
Poster 2.4.
Wijnand van der Velden
The “SeqR”, a Proprietary Non-antibody Scaffold that can Target Intrinsically Disordered Regions in GPCRs
Poster 2.5.
Florian Bößl
Unlocking the Activation Mechanism of Odorant Receptors through Large-Scale MD Simulations
Poster 2.6.
Jaume Lillo
Harnessing Cannabidiol to Reshape Microglial Response and Enhance Neuronal Survival in a Neonatal Hypoxia-Ischemia Model
Poster 2.7.
Camilla Guccione
Computational Insight into Small Molecule Binding to Gastrin- Releasing Peptide Receptor
Poster presentations will be live-streamed on November 26, 2024 from 15:50 to 16:20 CET.
Poster 3.2.
Kristoffer Sahlholm
Estimation of Dopamine D1 Receptor Agonist Binding Kinetics Using Time-Resolved Functional Assays
Poster 3.3.
Maris-Johanna Tahk
Quantifying Fluorescent Ligand Internalisation with High Content Imaging Techniques
Poster 3.5.
Matteo Pavan
Rational Design of Novel Positive Allosteric Modulators (PAMs) of the A3 Adenosine Receptor through the ‘Lipid Trolling’ Strategy
Poster 3.6.
Tomasz Stepniewski
An arginine switch drives the stepwise activation of β-arrestin
Poster 3.7.
Julie Delaroche
Split-NanoBiT-BRET-based Biosensors as tools to Query Mitochondrial GPCRs Localization
Poster 3.8.
Marija Popović-Nikolić
Understanding the ionization pattern of bilastine, histamine H1 receptor antagonist
Poster presentations will be live-streamed on November 26, 2024 from 18:50 to 19:20 CET.
Poster 4.1.
Clizia Russotto
Discovery of non-peptide ligands targeting the human Gonadotropin-Releasing Hormone Receptor
Poster 4.2
Francesco Fontanive
P2Y12 receptor goes towards activation: insights by Principal Component Analysis
Poster 4.3.
Aleix Quintana
Structure-based design of serotonin 5-HT2C receptor positive allosteric modulators for the treatment of obesity
Poster 4.4.
Marta López Balastegui
A ML-based approach for predicting variant impact on GPCR function
Poster 4.5.
Alejandro Peralta-García
Simulating the GPCRome: Large-scale analysis of AI-predicted and state-specific GPCR structures
Poster 4.7.
Anna Grimm
Cryo-EM structures of GPCR complexes obtained by rationalized cell-free production pipelines
Poster 4.8.
Marija Čarapić
Sensitive and simple UHPLC-MS/MS method for simultaneous determination of purity and assay of antipsychotic drug ziprasidone
Poster presentations will be live-streamed on November 27, 2024 from 11:30 to 12:00 CET.
Poster 5.2.
Shubham Vishnoi
Computational Design of Therapeutic Peptides Targeting Triple GPCR Agonist Activity
Poster 5.3.
Judith Alenfelder
Chemogenetic G protein-ligand pairs for causal investigation of cellular biology in vitro and in vivo
Poster 5.4.
Lucía González-Pico
Disrupting the adenosine axis in cancer immunotherapy: N-substituted pyrimidine derivatives to access A2B and dual A2A/A2B ligands
Poster 5.5.
Owen Underwood
ModuMelt™: Allosteric Modulator hit confirmation and characterisation
Poster 5.6.
Joan Biel Rebassa Palou
The impact of the CB1R-OX1R heteromeric complex on Alzheimer's disease
Poster 5.7.
Estefanía Moreno
Design of small non-peptidic ligands that alter heteromerization between cannabinoid CB1 and serotonin 5HT2A receptors
Poster 5.8.
Christian Lombo
Correlating Structure-activity Relationship analysis with luminescence assays in living cells to improve muscarinic M1-selective bitopic ligands
Poster presentations will be live-streamed on November 27, 2024 from 15:10 to 15:40 CET.
Poster 6.2.
Charlotte Crauwels
GPCRchimeraDB: a database to support the design of novel chimeric G-Protein Coupled Receptors for structure elucidation, ligand discovery and pathway understanding.
Poster 6.3.
Hongyue Liu
Structural mass spectrometry captures residue-resolved comprehensive conformational rearrangements of a G protein-coupled receptor
Poster 6.4.
Anna Chorianopoulou
Hit-to-Lead Optimization of Heterocyclic Carbonyloxycarboximidamides as Selective Antagonists at Human Adenosine A3 Receptor
Poster 6.5.
David Shi
Complex formation of cell-free synthesized short chain fatty acid receptors
Poster 6.7.
Shanshan Li
Profiling the GPCRome in Mouse Brain of Mental Disease Models Using a Comprehensive Spectral Library
Poster 6.8.
Antonio Capó Quetglas
Heteromeric Interaction Between Adenosine A2A and Cannabinoid CB2 Receptors in Stroke: A Promising Therapeutic Target to Enhance Microglial Neuroprotective Responses